掌握药物代谢的主要途径、部位 熟悉主要药物代谢酶—混合功能氧化酶的性质和代谢条件 熟悉影响药物代谢的因素 了解运用药物代谢酶性质进行制剂设计的方法 I. Introduction II. Drug Metabolism Enzyme & Site III. First Pass Effect & Hepatic Extraction IV. Metabolism Reaction V. Effects on Drug Metabolism VI. Drug Metabolism & Preparation Design VII.Study Technique(了解)
I. Overview of Regulation 8.1 Major modes of regulation II. Regulation of Enzyme Activity (Posttranslational level regulation) 8.2 Noncovalent enzyme inhibition 酶活的非共价抑制 8.3 Covalent Modification of Enzyme 酶的共价修饰 III. DNA-Binding Proteins and Regulation of Transcription by Negative and Positive Control (Transcriptional level regulation) 转录水平调控