复旦大学:《药物设计学》课程教学资源(虚拟实验室课外实践)Exercises for Drug Design Courses_Practice-III-4E MEDICINAL CHEMISTRY AND MOLECULAR MODELING:AN INTEGRATION FOR THE TEACHING OF DRUG STRUCTURE–ACTIVITY RELATIONSHIP AND THE MOLECULAR BASIS OF DRUG ACTION
复旦大学:《药物设计学》课程教学资源(虚拟实验室课外实践)Exercises for Drug Design Courses_Practice-III-2E A LABORATORY COURSE IN MEDICINAL CHEMISTRY INTRODUCING MOLECULAR MODELING
筛选途径需要解决的基本问题 I. 结构多样性(Diversity) II. 转化医学(Translational Medicine, from bench to bedside) 合成化合物的筛选 组合化学、多样性导向合成及片段库 转化医学 (Translational Medicine, from bench to bedside, from bed to bench) Neoclassic drug discovery 新经典药物发现 —— Phenotypic Screening